Mal-Dap(Boc)-OPfp

Synonyms
2,3,4,5,6‐pentafluorophenyl (2S)‐3‐{[(tert‐butoxy)carbonyl]amino}‐2‐(2,5‐dioxo‐2,5‐dihydro‐1H‐pyrrol‐1‐yl)propanoate

ID

ET-157

Formula

C18H15F5N2O6

CAS

1887132-90-2

MW

450.3

Purity

>98%

Storage

+2 ... +8 °C

Product image

References

Mal-Dap(Boc)-OPfp is used in drug conjugate construction leading to more stable conjugates due to Dap neighbouring-group assistance. This strategy is widely used by Seattle Genetics and others. Lyon et al PCT Int. Appl. (2015), WO 2015057699 A2; Cong et al PCT Int. Appl. (2017), WO 2017196598 A1; Burke et al PCT Int. Appl. (2017), WO 2017096311 A1.

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